Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6364 |
Desfesoterodine
5-HMT,(R)-5-Hydroxymethyl Tolterodine,(R)-5-羟甲基托特罗定,PNU-200577,5-HM,5-hydroxymethyl Tolterodine |
AChR | Neuroscience |
Desfesoterodine (5-HMT) 是选择性毒蕈碱受体拮抗剂,Kb 和pA2分别为 0.84 nM 和 9.14。它可改善大鼠脑梗死诱导膀胱过度活动,是 Tolterodine 和 Fesoterodine 的主要药理活性代谢产物。 | |||
T6364L |
Desfesoterodine fumarate
PNU-200577 fumarate,UNII-607O3D83YQ |
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Desfesoterodine fumarate is a bio-active chemical. Detailed information has not been published. |