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Cat. No. | Product Name | Target | Signaling Pathways |
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T81445 |
PKRA83 hydrochloride hydrate
PKRA7 hydrochloride hydrate |
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PKRA83 hydrochloride hydrate是一种高效的促动力拮抗剂,与PK2及其受体PKR1和PKR2进行竞争性结合。该化合物在抑制PK2受体方面表现出色,其对PKR1和PKR2的IC50值分别为5.0 nM和8.2 nM。此外,PKRA83 hydrochloride hydrate还具备抗癌、抗关节炎以及抗血管生成的活性,并能够穿透血脑屏障。 | |||
T63446 |
PKRA83
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PKRA83 是一种能够透过血脑屏障的 potent prokineticin (PK2) 拮抗剂,可竞争 PK2 与其受体 PKR1 和 PKR2 的结合。PKRA83 能够有效抑制 PK2 受体,可作用于 PKR1 (IC50: 5.0 nM) 和 PKR2 (IC50: 8.2 nM)。PKRA83 表现出抗癌和抗血管生成作用。 |
Cat. No. | Product Name | Species | Expression System |
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TMPY-03656 |
PRKAR1A Protein, Human, Recombinant (His)
PRKAR1,CAR,CNC1,PPNAD1,CNC,protei... |
Human | HEK293 Cells |
PRKAR1A Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 36.2 kDa and the accession number is P10644. |