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Cat. No. Product Name Target Signaling Pathways
TP1955 PKC β pseudosubstrate

Selective cell-permeable peptide inhibitor of protein kinase C (IC50 ~ 0.5 μM). Consists of amino acids 19 - 31 of PKC pseudosubstrate domain linked by a disulphide bridge to a cell permeabilisation Antennapedia domain vector peptide. The Antennapedia pep
TP1955L PKC β pseudosubstrate acetate

PKC β pseudosubstrate醋酸盐,Protein kinase C beta pseudosubstrate,PKC beta pseudosubstrate,PKC β pseudosubstrate acetate (172308-76-8 Free base)

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
PKC β pseudosubstrate acetate (PKC β pseudosubstrate acetate (172308-76-8 Free base)) 是一种选择性的、细胞渗透的 PKC 抑制剂。
TP1956L PKC ζ pseudosubstrate acetate

PKC ζ pseudosubstrate acetate (799764-07-1 free base)

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
PKC ζ pseudosubstrate acetate 是蛋白激酶 C (PKC) ζ 的抑制剂;附着于细胞通透性触角足结构域载体肽。由 PKC ζ 假底物结构域的氨基酸 113-129 组成,通过二硫键连接到触角足结构域载体肽。 Antennapedia 肽在 4 或 37°C 时被完整细胞积极吸收,确保快速有效地吸收抑制肽。一旦进入细胞,二硫键在细胞质中被还原,导致抑制肽的释放。通过 PKC ζ 非依赖性途径诱导肥大细胞脱粒。
T75885 PKC β pseudosubstrate TFA

PKCβ pseudosubstrate TFA 是一种选择性的、细胞渗透的 PKC 抑制剂。
T80071 PKCζ/ι pseudosubstrate inhibitor

PKCζ/ι偽基質抑制劑對PKC酶家族表現廣譜抑制作用,並可能促成記憶功能障礙。
T80508 PKCη pseudosubstrate inhibitor,myristoylated

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
Myristoylated PKCη pseudosubstrate inhibitor 是一种具有细胞渗透性的化合物,它主要应用于研究PKCη的作用机制。
T80507 PKCθ pseudosubstrate peptide inhibitor,myristoylated

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
Myristoylated PKCθ pseudosubstrate peptide inhibitor 是一款合成肽,专门用于研究 PKCθ 的机制。

化合物

PKC β pseudosubstrate
Cat.No: TP1955
Synonym:
Target:
PKC β pseudosubstrate acetate
Cat.No: TP1955L
Synonym: PKC β pseudosubstrate醋酸盐,Protein kinase C beta pseudosubstrate,PKC beta pseudosubstrate,PKC β pseudosubstrate acetate (172308-76-8 Free base)
Target: PKC
PKC ζ pseudosubstrate acetate
Cat.No: TP1956L
Synonym: PKC ζ pseudosubstrate acetate (799764-07-1 free base)
Target: PKC
PKC β pseudosubstrate TFA
Cat.No: T75885
Synonym:
Target:
PKCζ/ι pseudosubstrate inhibitor
Cat.No: T80071
Synonym:
Target:
PKCη pseudosubstrate inhibitor,myristoylated
Cat.No: T80508
Synonym:
Target: PKC
PKCθ pseudosubstrate peptide inhibitor,myristoylated
Cat.No: T80507
Synonym:
Target: PKC
TargetMol Loading
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