Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP1952L |
PG 106 acetate
PG 106 acetate(944111-22-2 Free base) |
Melanocortin Receptor | GPCR/G Protein; Neuroscience |
PG 106 acetate 是一种有效的特异性人黑皮质素 3 (hMC3) 受体拮抗剂,IC50 为 210 nM。 PG 106 acetate 对 hMC5 受体和 hMC4 受体没有活性,hMC4 受体的 EC50 为 9900 nM。 | |||
TP1952 |
PG106
PG 106 |
||
Selective hMC3 receptor antagonist (IC50 = 210 nM). Exhibits no activity at hMC4 receptors and hMC5 receptors. |