Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T12428L |
PF-06726304
|
Histone Methyltransferase | Chromatin/Epigenetic |
PF-06726304 是选择性EZH2有效抑制剂,具有强抗肿瘤生长活性。它抑制野生型和 Y641N 突变型 EZH2,Ki 分别为 0.7 和 3.0 nM。 | |||
T12428 |
PF-06726304 acetate
|
Histone Methyltransferase | Chromatin/Epigenetic |
PF-06726304 acetate is a selective inhibitor of EZH2, with robust antitumor growth activity. |