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Cat. No. Product Name Target Signaling Pathways
T8711 PF-05186462

PF-05150122

Sodium Channel Membrane transporter/Ion channel
PF-05186462 (PF-05150122)是选择性的人Nav1.7电压依赖性钠通道抑制剂,IC50为 21 nM,与其他钠通道 (Nav 1.1、1.2、1.3、1.4、1.5、1.6 和 1.8) 相比,它对 Nav1.7显示出显著的选择性。PF-05186462在急性或慢性疼痛中具有研究价值。
T71166 PF-05150122

PF-05150122 is a novel potent and selective human Nav1.7 blocker.
T71164 CXN37378

CXN37378, also known as NAP, is a potent and selective antagonist for the μ-opioid receptor (MOR). This product has no formal name at the moment. For the convenience of communication, a temporary code name was therefore proposed according to MedKoo Chemical Nomenclature (see web page: https://www.medkoo.com/page/naming).

化合物

PF-05186462
Cat.No: T8711
Synonym: PF-05150122
Target: Sodium Channel
PF-05150122
Cat.No: T71166
Synonym:
Target:
CXN37378
Cat.No: T71164
Synonym:
Target:
TargetMol Loading
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