Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T71166 |
PF-05150122
|
||
PF-05150122 is a novel potent and selective human Nav1.7 blocker. | |||
T8711 |
PF-05186462
PF-05150122 |
Sodium Channel | Membrane transporter/Ion channel |
PF-05186462 (PF-05150122)是选择性的人Nav1.7电压依赖性钠通道抑制剂,IC50为 21 nM,与其他钠通道 (Nav 1.1、1.2、1.3、1.4、1.5、1.6 和 1.8) 相比,它对 Nav1.7显示出显著的选择性。PF-05186462在急性或慢性疼痛中具有研究价值。 | |||
T71164 | CXN37378 | ||
CXN37378, also known as NAP, is a potent and selective antagonist for the μ-opioid receptor (MOR). This product has no formal name at the moment. For the convenience of communication, a temporary code name was therefore proposed according to MedKoo Chemical Nomenclature (see web page: https://www.medkoo.com/page/naming). |