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Cat. No. Product Name Target Signaling Pathways
T12394 PDE5-IN-2

PDE Metabolism
PDE5-IN-2 is a potent, highly selective, and orally active inhibitor of PDE5(IC50 of 0.31 nM)
T37325 Lodenafil carbonate

Lodenafil carbonate, a prodrug dimer that delivers Lodenafil in vivo, is an orally active inhibitor of phosphodiesterase type 5 (PDE5), indicated for the treatment of erectile dysfunction (ED)[1][2].
T79533 PDE5-IN-10

PDE5-IN-10 (compound 4b),一有效PDE5抑制剂,IC50值为20 nM。该化合物体外微粒体稳定性增强(t1/2= 44.6 分钟),在长期增强恢复方面效果显著,适用于阿尔茨海默病(AD)研究。

化合物

PDE5-IN-2
Cat.No: T12394
Synonym:
Target: PDE
Lodenafil carbonate
Cat.No: T37325
Synonym:
Target:
PDE5-IN-10
Cat.No: T79533
Synonym:
Target:
TargetMol Loading
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