Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T30188L |
Atagabalin HCl
PD-0200390 HCl,Atagabalin HCl(223445-75-8 Free base) |
Calcium Channel | Membrane transporter/Ion channel; Metabolism |
Atagabalin HCl 是一种新型电压依赖性钙通道(VDCC)α2δ亚基(1 和 2)配体,会影响慢波睡眠,可用于治疗失眠。 | |||
T30188 |
Atagabalin
PD 0200390,PD-0200390,PD0200390 |
||
Atagabalin, also known as PD 0200390, is a gabamimetic agent under development for the treatment for insomnia. Atagabalin is related to gabapentin, which similarly binds to the α2δ calcium channels (1 and 2). It was discontinued following unsatisfactory t | |||
T30188L1 |
(Iso)-Atagabalin HCl
(Iso)-Atagabalin HCl((Iso)-223445-75-8) |
Others | Others |
(Iso)-Atagabalin HCl(isomer-Atagabalin HCl) 是一种可用于治疗非恢复性睡眠的α -2- δ配体。 |