Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T60157 |
PBRM1-BD2-IN-8
|
Epigenetic Reader Domain | Chromatin/Epigenetic |
PBRM1-BD2-IN-8 (compound 34) 是一种强效的 PBRM1 Bromodomain 抑制剂 (PBRM1-BD2 Kd=4.4 μM, PBRM1-BD2 IC50=0.16 μM; PBRM1-BD5 Kd=25 μM),其具有抗癌活性。 |