Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TQ0179 |
PAP-1
5-(4-Phenoxybutoxy)psoralen |
Potassium Channel | Membrane transporter/Ion channel |
PAP-1 (5-(4-Phenoxybutoxy)psoralen) 是口服活性的Kv1.3选择性阻滞剂 (EC50=2 nM)。它依赖性阻止 Kv1.3,并优先与通道的 C 型失活状态结合来发挥作用。 |