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Cat. No. Product Name Target Signaling Pathways
TP1139 Orexin B, human

Human orexin B

Orexin B, human is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively. Orexin B is a hypothalamatic neuropeptide stimulating food intake in rats.
TP1138 Orexin B, human TFA (205640-91-1 free base)

Orexin B, human TFA,Human orexin B TFA

Orexin B, human (TFA) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2.
TP1975 [Ala11,D-Leu15]-Orexin B(human)

[Ala11,D-Leu15]-Orexin B

Highly potent and selective OX2 receptor agonist; displays 400-fold selectivity over OX1 receptors. EC50 values are 0.13 and 52 nM for human OX2 and OX1 receptors respectively.
T75920 Orexin B, human TFA

Orexin B, human (TFA) 是 Orexin 受体的内源性激动剂,与 OX1和 OX2结合的 Ki 值分别为 420 和 36 nM。
T75921 [Ala11,D-Leu15]-Orexin B(human) TFA

[Ala11,D-Leu15]-Orexin B(human) TFA为高效的orexin-2 receptor (OX2)选择性激动剂。其对OX2展现出比OX1 (52 nM) 高达400倍的较高选择性(EC50=0.13 nM)。

化合物

Orexin B, human
Cat.No: TP1139
Synonym: Human orexin B
Target:
Orexin B, human TFA (205640-91-1 free base)
Cat.No: TP1138
Synonym: Orexin B, human TFA,Human orexin B TFA
Target:
[Ala11,D-Leu15]-Orexin B(human)
Cat.No: TP1975
Synonym: [Ala11,D-Leu15]-Orexin B
Target:
Orexin B, human TFA
Cat.No: T75920
Synonym:
Target:
[Ala11,D-Leu15]-Orexin B(human) TFA
Cat.No: T75921
Synonym:
Target:
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