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Cat. No. | Product Name | Target | Signaling Pathways |
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T38470 |
Obestatin (human)
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Obestatin (human) 是一种由 preproghrelin 经过剪切形成的G蛋白欧联实体39的内源性配体,可以剂量依赖的方式抑制进食,可用于研究肥胖。 | |||
TP2279L |
Obestatin (rat) acetate
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GHSR | GPCR/G Protein |
Obestatin (rat) acetate 是 G 蛋白偶联受体 39 (GPR39) 的内源性配体。它具有抗炎、抗心肌梗塞和抗氧化特性。 它抑制食物摄入,抑制空肠收缩,并减少体重增加。 | |||
TP2279 |
Obestatin(rat)
Obestatin (rat) |
Others | Others |
Endogenous peptide that suppresses food intake and body weight-gain | |||
T35787 |
Obestatin (human) (trifluoroacetate salt)
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Obestatin is a 23 amino acid peptide hormone with a conserved C-terminal glycine residue and amidation site that is formed by cleavage of the ghrelin and obestatin prepropeptide.1It binds to the orphan receptor GPR39 (Kd= 1 nM) and stimulates cAMP production in CHO and HEK293 cells overexpressing human GPR39. Obestatin inhibits contraction of isolated mouse jejunum muscle strips induced by ghrelin .In vivo, obestatin (12.5-1,000 nmol/kg) suppresses food intake in a time- and dose-dependent manne... | |||
T81625 |
Obestatin(human) TFA
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Obestatin(human) TFA, 同源于与ghrelin相同的前体多肽,是一种内源性肽。该化合物抑制大鼠食欲并降低体重增加。 | |||
T75901 |
Obestatin(rat) TFA
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Obestatin(rat) TFA 是一个包含23个氨基酸的肽,由Ghrelin基因编码。该化合物能够抑制食欲和空肠收缩,并能减缓体重增加。同时,Obestatin(rat) TFA 作为G 蛋白偶联受体 39 (GPR39) 的内源性配体,发挥抗炎、抗心肌梗塞和抗氧化功能。 | |||
T81626 |
Obestatin(11-23)mouse, rat
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Obestatin(11-23)mouse, rat 是多肽,涉及能量平衡调节,抑制摄食。该化合物能使啮齿类动物食量减少、体重降低、及空肠收缩。 |
Cat. No. | Product Name | Target | Signaling Pathways |
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T4588 |
Glycochenodeoxycholic Acid
甘氨鹅脱氧胆酸,Glycine chenodeoxycholate,Chenodeoxycholylglycine,GCDCA,Glycochenodeoxycholate,Lithocholylglycine |
Apoptosis; Endogenous Metabolite | Apoptosis; Metabolism |
Glycochenodeoxycholic Acid (Lithocholylglycine) 是一种从脱氧鹅胆酸和甘氨酸在肝脏中形成的胆汁盐,可诱导肝细胞凋亡。它有洗涤剂的作用,可溶解脂肪吸收,并本身被吸收。 |