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抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T37668 CAY10448

CAY10448

Capsaicin is the primary active component of the heat and pain-eliciting lipid soluble fraction of the Capsicum pepper. Capsaicin signals are transduced by a heat-activated ion channel, the vanilloid receptor 1 (VR1), or transient receptor potential vanilloid 1 (TRPV1). CAY10448 is an iodinated nonivamide, a potent capsaicin receptor antagonist with an IC50 value of approximately 10 nM.
T1309 Propylthiouracil

丙硫氧嘧啶,Pseudocapsaicin,NSC 6498,丙基硫氧嘧啶,NSC 70461,6-n-Propylthiouracil,6-Propyl-2-thiouracil

Thyroid hormone receptor(THR) Endocrinology/Hormones
Propylthiouracil (6-n-Propylthiouracil) 是一种甲状腺过氧化物酶抑制剂,也是一种5'-脱碘酶抑制剂。

化合物

CAY10448
Cat.No: T37668
Synonym: CAY10448
Target:
Propylthiouracil
Cat.No: T1309
Synonym: 丙硫氧嘧啶,Pseudocapsaicin,NSC 6498,丙基硫氧嘧啶,NSC 70461,6-n-Propylthiouracil,6-Propyl-2-thiouracil
Target: Thyroid hormone receptor(THR)
Cat. No. Product Name Target Signaling Pathways
T1321 Nonivamide

Nonanoic acid vanillylamide,Pelargonic acid vanillylamide,辣椒素,Vanillyl-N-nonylamide,Pseudocapsaicin

TRP/TRPV Channel Membrane transporter/Ion channel
Nonivamide (Nonanoic acid vanillylamide) 具有激动活性,在静态毒性检测中,4d-EC50为 5.1 mg/L。

天然产物

Nonivamide
Cat.No: T1321
Synonym: Nonanoic acid vanillylamide,Pelargonic acid vanillylamide,辣椒素,Vanillyl-N-nonylamide,Pseudocapsaicin
Target: TRP/TRPV Channel
TargetMol Loading
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