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抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T50111 6-Fluorotryptamine hydrochloride

Others Others
6-Fluorotryptamine hydrochloride 是一种用作分子结构单元的化合物,是天然色胺生物碱血清素的衍生物。它是5-HT2A 和5-HT2C 血清素受体的激动剂,使其成为开发治疗各种精神和神经疾病的新药的潜在候选者。
T4615 Balsalazide sodium hydrate

巴柳氮钠水合物,Balsalazide disodium dihydrate,巴柳氮钠,Balsalazide disodium salt dihydrate,Balsalazide disodium

STAT; Interleukin Immunology/Inflammation; JAK/STAT signaling; Stem Cells
Balsalazide sodium hydrate (Balsalazide disodium) 可通过调节IL-6/STAT3通路起抑癌作用,可用于治疗炎症性肠病。
T38192 Unifiram

Others Others
Unifiram 是一种认知增强剂。 Unifiram 诱导大鼠海马 CA1 区场兴奋性突触后电位 (fEPSP) 幅度的持久增加 (EC50= 27 nM) 并增加大鼠大脑皮层中乙酰胆碱 (ACh) 的释放。

化合物

6-Fluorotryptamine hydrochloride
Cat.No: T50111
Synonym:
Target: Others
Balsalazide sodium hydrate
Cat.No: T4615
Synonym: 巴柳氮钠水合物,Balsalazide disodium dihydrate,巴柳氮钠,Balsalazide disodium salt dihydrate,Balsalazide disodium
Target: STAT, Interleukin
Unifiram
Cat.No: T38192
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
TN6407 New compound 5

New compound 5是一种天然产物,属于五味子科五味子属,其产品编号为 TN6407。New compound 5可用作对照参考。
T37690 Phenylpyropene A

Phenylpyropene A is a fungal metabolite originally isolated from P. griseofulvum that has enzyme inhibitory and insecticidal activities.1,2,3 It inhibits acyl-coenzyme A:cholesterol acyltransferase (ACAT; IC50 = 0.8 μM).1 Phenylpyropene A inhibits diacylglycerol acyltransferase (DGAT) in rat liver microsomes (IC50 = 78.7 μM). It induces mortality in 100% of M. persicae when used at a concentration of 5 ppm.3 |1. Kwon, O.E., Rho, M.C., Song, H.Y., et al. Phenylpyropene A and B, new inhibitors of ...

天然产物

New compound 5
Cat.No: TN6407
Synonym:
Target:
Phenylpyropene A
Cat.No: T37690
Synonym:
Target:
TargetMol Loading
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