搜索结果

Search Results for " netupitant "

如果没找到您满意的产品或者您对产品有其他要求，可以联系我们专业顾问为您提供针对性的合理建议。 QQ咨询网站留言咨询

Cat. No.	Product Name	Target	Signaling Pathways
T6905	Netupitant Ro 67-31898/000,奈妥吡坦,CID 6451149	Neurokinin receptor	GPCR/G Protein; Neuroscience
	Netupitant (CID 6451149) 是一种高效选择性、可口服的神经激肽 1 受体 (NK1) 拮抗剂，具有止吐作用，在 CHO 细胞中对 hNK1的 Ki 值为 0.95 nM。
T12212	Netupitant metabolite N-desmethyl Netupitant N-desmethyl Netupitant	Others	Others
	N-desmethyl Netupitant is a highly selective antagonist of NK1 receptor, and is Netupitant metabolite.
T12211	Netupitant metabolite Monohydroxy Netupitant Monohydroxy Netupitant	Others	Others
	Monohydroxy Netupitant is a highly selective antagonist of NK1 receptor, and is Netupitant metabolite.
T12213	Netupitant metabolite Netupitant N-oxide Netupitant N-oxide	Others	Others
	Netupitant N-oxide is a highly selective antagonist of NK1 receptor, is Netupitant metabolite.
T12210	Netupitant D6 CID-6451149 D6	Others	Others
	Netupitant D6 is the deuterium labeled Netupitant, which is a selective and orally active antagonist of neurokinin-1 receptor.
T19434	Monohydroxy Netupitant D6	Others	Others
	Monohydroxy Netupitant D6 is a metabolite of Netupitant.
T19474	Netupitant N-oxide D6	Others	Others
	Netupitant N-oxide D6 is a Netupitant metabolite, is the deuterium labeled Netupitant N-oxide.
T19452	N-desmethyl Netupitant D6	Others	Others
	N-desmethyl Netupitant D6 is the deuterium labeled N-desmethyl Netupitant, which is a Netupitant metabolite.
T15341	Fosnetupitant Pronetupitant	Others	Others
	Fosnetupitant is a methylene phosphate prodrug of Netupitant. It has a pKi of 9.5 for the human NK1 receptor.
T78104	Fosnetupitant chloride monohydrochloride Pronetupitant chloride monohydrochloride	Neurokinin receptor	GPCR/G Protein; Neuroscience
	Fosnetupitant chloride monohydrochloride（Pronetupitant chloride monohydrochloride）为NK1受体拮抗剂，对人NK1受体和NK3受体的pKi分别为9.5和6.1。它是奈妥匹坦的亚甲基磷酸酯前体。
T9735	6-(4-methylpiperazin-1-yl)-4-o-tolylnicotinamide	Others	Others
	6-(4-methylpiperazin-1-yl)-4-o-tolylnicotinamide 可用于合成befetupitant 和netupitant。