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Targets Recommended: Phosphatase

10

抑制剂 & 化合物

2

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T79622 h-NTPDase-IN-3

Phosphatase Metabolism
h-NTPDase-IN-3 是一种 h-NTPDase 抑制剂,抑制 h-NTPDase1,h-NTPDase2,h-NTPDase3 和 h-NTPDase8。
T77661 h-NTPDase-IN-4

Phosphatase Metabolism
h-NTPDase-IN-4 是 NTPDase 的泛抑制剂,对 h-NTPDase1, 1h-NTPDase2, h-NTPDase3, h-NTPDase8具有抑制作用,IC50 分别为 3.58 μM , 10.21 μM , 0.13 μM , 13.57 μM 。
T14320 ARL67156 trisodium salt

Others Others
ARL 67156 is a weak competitive inhibitor of NTPDase1 (CD39), NTPDase3 and NPP1, with Kis of 11, 18 and 12 μM, respectively[1]. ARL67156 trisodium salt is an inhibitor of ecto-ATPase.
T62633 NTPDase-IN-3

NTPDase-IN-3 (Compound 5e) 是一种 NTPDase 抑制剂,IC50值分别为 0.38 μM (NTPDase3), 0.05 μM (NTPDase8), 0.21 μM (NTPDase1), 1.07 μM (NTPDase2)。NTPDase-IN-3 可用于癌症和血栓形成的研究。
T73644 ARL67156 trisodium hydrate

ARL67156 (FPL 67156) trisodium hydrate 是一种ecto-ATPase 抑制剂。ARL67156 trisodium hydrate 是竞争性 NTPDase1 (CD39),NTPDase3 和 NPP1 抑制剂,Ki 分别为 1118 和 12 μM。ARL67156 trisodium hydrate 可用于钙化性主动脉瓣疾病、哮喘等疾病的研究。
T79623 h-NTPDase-IN-5

Phosphatase Metabolism
h-NTPDase-IN-5(化合物3b)是一种NTPDase的泛抑制剂,其IC50s对于h-NTPDase11.10 μM,h-NTPDase2为44.73 μM,h-NTPDase3为26.14 μM,h-NTPDase8为0.32 μM。
T12519 Sodium metatungstate

POM-1,聚钨酸钠,Sodium polyoxotungstate

Phosphatase Metabolism
Sodium metatungstate (Sodium polyoxotungstate) 是一种外核苷三磷酸二磷酸水解酶抑制剂,能够抑制 ATP 的分解,并阻断中枢突触传递,这是独立于抑制 NTPDase 而发挥作用的。
T79491 h-NTPDase-IN-1

Phosphatase Metabolism
h-NTPDase-IN-1 (Compound 3i) 是一种针对 h-NTPDase 的抑制剂,对 h-NTPDase1 和 h-NTPDase3 的抑制作用表现在 IC50 值分别为 2.88 μM 和 0.72 μM。该化合物在血栓、炎症、糖尿病及癌症研究领域有潜在应用。
T73645 ARL67156 triethylamine

ARL67156 (FPL 67156) triethylamine 是一种ecto-ATPase 抑制剂。ARL67156 triethylamine 是竞争性 NTPDase1 (CD39),NTPDase3 和 NPP1 抑制剂,Ki 分别为 1118 和 12 μM。ARL67156 triethylamine 可用于钙化性主动脉瓣疾病、哮喘等疾病的研究。
T79607 h-NTPDase-IN-2

hNTPDase-IN-2

Phosphatase Metabolism
h-NTPDase-IN-2 是一种广谱 NTPDase 抑制剂,对多种 h-NTPDas 亚型都具有抑制作用。

化合物

h-NTPDase-IN-3
Cat.No: T79622
Synonym:
Target: Phosphatase
h-NTPDase-IN-4
Cat.No: T77661
Synonym:
Target: Phosphatase
ARL67156 trisodium salt
Cat.No: T14320
Synonym:
Target: Others
NTPDase-IN-3
Cat.No: T62633
Synonym:
Target:
ARL67156 trisodium hydrate
Cat.No: T73644
Synonym:
Target:
h-NTPDase-IN-5
Cat.No: T79623
Synonym:
Target: Phosphatase
Sodium metatungstate
Cat.No: T12519
Synonym: POM-1,聚钨酸钠,Sodium polyoxotungstate
Target: Phosphatase
h-NTPDase-IN-1
Cat.No: T79491
Synonym:
Target: Phosphatase
ARL67156 triethylamine
Cat.No: T73645
Synonym:
Target:
h-NTPDase-IN-2
Cat.No: T79607
Synonym: hNTPDase-IN-2
Target: Phosphatase
Cat. No. Product Name Species Expression System
TMPH-03284 CD39 Protein, Rat, Recombinant (E. coli, His)

Entpd1,ATP-DPH,Ecto-ATP diphosphohydrolase 1

Rat E. coli
In the nervous system, could hydrolyze ATP and other nucleotides to regulate purinergic neurotransmission. Could also be implicated in the prevention of platelet aggregation by hydrolyzing platelet-activating ADP to AMP. Hydrolyzes ATP and ADP equally well.
TMPH-03283 CD39 Protein, Rat, Recombinant (His)

ATP diphosphohydrolase,Entpd1,Nucleoside triphospha...

Rat Baculovirus Insect Cells
In the nervous system, could hydrolyze ATP and other nucleotides to regulate purinergic neurotransmission. Could also be implicated in the prevention of platelet aggregation by hydrolyzing platelet-activating ADP to AMP. Hydrolyzes ATP and ADP equally well.

重组蛋白

CD39 Protein, Rat, Recombinant (E. coli, His)
Cat.No: TMPH-03284
Species: Rat
Expression System: E. coli
CD39 Protein, Rat, Recombinant (His)
Cat.No: TMPH-03283
Species: Rat
Expression System: Baculovirus Insect Cells
TargetMol Loading
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