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Search Results for " nf-κb-in-13 "

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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T79999 NF-κB-IN-13

NF-κB NF-κB
NF-κB-IN-13(compound 12)在RAW264.7巨噬细胞中显著抑制了LPS诱导的NF-κB激活以及NO生成,表现出其抗炎效果。
T35406 α-MSH TFA

α-Melanocyte-stimulating hormone (α-MSH) is a 13-amino acid peptide hormone produced by post-translational processing of proopiomelanocortin (POMC) in the pituitary gland, as well as in keratinocytes, astrocytes, monocytes, and gastrointestinal cells.1It is an agonist of melanocortin receptor 3 (MC3R) and MC4R that induces cAMP production in Hepa cells expressing the human receptors (EC50s = 0.16 and 56 nM, respectively).2α-MSH (100 pM) reducesS. aureuscolony formation andC. albicansgerm tube fo...

化合物

NF-κB-IN-13
Cat.No: T79999
Synonym:
Target: NF-κB
α-MSH TFA
Cat.No: T35406
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T79962 Aloenin aglycone

Others Others
Aloenin aglycone (compound 13) 作为一种NF-κB抑制剂,可从芦荟渗出液中提取。它在抑制TNFα引发的NF-κB转录活性方面表现显著(IC50: 18.7 μM)。当HepG2细胞经10 ng/mL TNFα处理时,以10 μM Aloenin aglycone处理能有效下调诱导型一氧化氮合酶(iNOS)及细胞间粘附分子1(ICAM-1)的基因表达。

天然产物

Aloenin aglycone
Cat.No: T79962
Synonym:
Target: Others
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