Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7147 |
Valbenazine
NBI-98854 |
Monoamine Transporter | Membrane transporter/Ion channel |
Valbenazine (NBI-98854) 是一种高度选择性的囊泡单胺转运蛋白 2 (VMAT2) 抑制剂,Ki 为 110-190 nM,用于治疗迟发性运动障碍。 | |||
T71922 | MS2734 | ||
MS2734 is a novel Bisubstrate Inhibitor of Nicotinamide N-Methyltransferase (NNMT). | |||
T22452 |
Valbenazine tosylate
結苯那嗪,NBI-98854 |
Monoamine Transporter | Membrane transporter/Ion channel |
Valbenazine tosylate, the tosylate salt of valbenazine, is a vesicular monoamine transporter 2 (VMAT2) inhibitor with a Ki value of 150 nM while displaying no significant binding to VAMT1(Ki<10 μM). |