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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T16789 Rosoxacin

罗索沙星,Acrosoxacin

Antibacterial; Antibiotic Microbiology/Virology
Rosoxacin (Acrosoxacin) 是具有口服活性的喹诺酮类抗生素,具有广谱的抗菌活性,抑制革兰氏阴性菌,包括淋病奈瑟氏球菌(MIC90=0.03 mg/ml)。它在尿路感染中有应用的潜能。
T38290 Leucomycin A4

Leucomycin A4

Leucomycin A4 is a macrolide antibiotic that has been found in S. kitasatoensis. It is active against a variety of bacteria, including S. aureus, B. subtilis, C. diphtheriae, N. gonorrhoeae, and H. influenzae (MICs = 0.15, 1.25, 0.15, 0.6, and 0.15 μg/ml, respectively).
T83703 BLP-3 TFA

Bombin-like Peptide 3

BLP-3是一种在X. laevis皮肤中表达的内源性多肽,具有抗菌特性。在20 µg/ml的浓度下对N. meningitidis、N. gonorrhoeae、N. lactamica和N. cinerea有效。BLP-3折叠成α-螺旋结构,能插入并破坏类细菌膜。
T61481 TP0480066

TP0480066, a selective topoisomerase II inhibitor, demonstrates excellent inhibitory activity against DNA gyrase (IC50 = 1.10 nM) and topo IV (IC50 = 62.89 nM). This compound exhibits potent efficacy against multiple bacterial species, including drug-resistant strains. Moreover, TP0480066 displays significant inhibitory activity against N. gonorrhoeae, making it suitable for research on gonorrhea [1] [2].

化合物

Rosoxacin
Cat.No: T16789
Synonym: 罗索沙星,Acrosoxacin
Target: Antibacterial, Antibiotic
Leucomycin A4
Cat.No: T38290
Synonym: Leucomycin A4
Target:
BLP-3 TFA
Cat.No: T83703
Synonym: Bombin-like Peptide 3
Target:
TP0480066
Cat.No: T61481
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T0819 Spiramycin

Espiramicin,螺旋霉素,Sequamycin,Rovamycin,Provamycin,Formacidine

Antibacterial; Antibiotic; Parasite Microbiology/Virology
Spiramycin (Rovamycin) 是一种由安博链霉菌产生的大环内酯类抗生素,具有抗细菌和弓形虫活性,并具有抗寄生虫作用。它由 16 个内酯环组成,其上附着 mycaminose,forosamine 和 mycarose 三种糖。

天然产物

Spiramycin
Cat.No: T0819
Synonym: Espiramicin,螺旋霉素,Sequamycin,Rovamycin,Provamycin,Formacidine
Target: Antibacterial, Antibiotic, Parasite
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