Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T36061 |
N-Desmethyl Sildenafil
Desmethylsildenafil,UK-103,320 |
Drug Metabolite | Metabolism |
N-Desmethyl Sildenafil (UK-103,320) (Desmethylsildenafil) 是Sildenafil的主要代谢物,是一种强效的磷酸二酯酶类型5(PDE5)抑制剂。 | |||
T36062 | N-Desmethyl Sildenafil (citrate) | ||
N-Desmethyl sildenafil is a major metabolite of sildenafil . N-Desmethyl sildenafil is formed via oxidative metabolism of sildenafil by the cytochrome (CYP) P450 isoforms CYP3A4, CYP3A5, and CYP3A7. |