Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T19449 |
N-desmethyl Enzalutamide D6
N-desmethyl MDV 3100 D6 |
Androgen Receptor | Endocrinology/Hormones |
N-desmethyl Enzalutamide D6 is a deuterium labeled N-desmethyl Enzalutamide. | |||
T19450 |
N-desmethyl Enzalutamide
4-[3-[4-氰基-3-(三氟甲基)苯基]-5,5-二甲基-4-氧代-2-硫代-1-咪唑烷基]-2-氟苯甲酰胺,N-desmethyl MDV 3100 |
Androgen Receptor | Endocrinology/Hormones |
N-desmethyl Enzalutamide (N-desmethyl MDV 3100) 是一种 Enzalutamide 的主要活性代谢物,具有与 Enzalutamide 相似的一级和二级药效功效,并在与 Enzalutamide 大致相同的血浆浓度下循环。 |