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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T37548 azido-FTY720

azido-FTY720

FTY720 is a derivative of ISP-1 (myriocin), a fungal metabolite of the Chinese herb Iscaria sinclarii as well as a structural analog of sphingosine. It is a novel immune modulator that prolongs allograft transplant survival in numerous models by inhibiting lymphocyte emigration from lymphoid organs. FTY720 is phosphorylated by sphingosine kinase, which then acts as a potent agonist at four of the sphingosine-1-phosphate (S1P) receptors (S1P1, S1P3, S1P4, and S1P5). Down-regulation of S1P1 recept...

化合物

azido-FTY720
Cat.No: T37548
Synonym: azido-FTY720
Target:
Cat. No. Product Name Target Signaling Pathways
T16165 Myriocin

ISP-I,Thermozymocidin

HCV Protease; Antifungal Microbiology/Virology; Proteases/Proteasome
Myriocin (Thermozymocidin) 是一种从 Myriococcum albomyces 中得到的代谢产物,是一种丝氨酸-棕榈酰转移酶 (SPT) 抑制剂,具有潜在的抗肿瘤抗癌和抗寄生虫活性,通过 PI3K/Akt/mTOR 通路调节巨噬细胞极化和功能来抑制肿瘤生长。Myriocin 抑制 HCV 感染,可用于研究神经病变和真菌感染。

天然产物

Myriocin
Cat.No: T16165
Synonym: ISP-I,Thermozymocidin
Target: HCV Protease, Antifungal
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