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抑制剂 & 化合物

3

天然产物

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Cat. No. Product Name Target Signaling Pathways
T75304 Mupirocin calcium

Mupirocin (BRL-4910A, Pseudomonic acid) calcium 可从Pseudomonas fluorescens 中分离得到,是一种有口服活性的抗生素。Mupirocin calcium 通过可逆地抑制异亮氨酸转移 RNA,从而抑制细菌蛋白和 RNA 的合成而发挥抗菌作用。
T25997 Pseudomonic acid C

Mupirocin calcium impurity B

Pseudomonic acid C is the analogue of Pseudomonic Acid D which is an antibiotic agent from Pseudomonas fluorescens.
T14359 AVX 13616

Others Others
AVX 13616 shows the potent in vivo antibacterial activity of Avexa’s lead antibacterial candidate; particularly against drug-resistant Staphylococcus pathogens. IC50 value: 2-4 ug/ml (MICs) Target: antibacterial agent AVX13616 was as active as mupirocin i

化合物

Mupirocin calcium
Cat.No: T75304
Synonym:
Target:
Pseudomonic acid C
Cat.No: T25997
Synonym: Mupirocin calcium impurity B
Target:
AVX 13616
Cat.No: T14359
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T1465 Mupirocin

Pseudomonic acid,莫匹罗星,BRL-4910A

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Mupirocin (BRL-4910A) 是从Pseudomonas fluorescens 中分离得到的一种有口服活性的抗生素。它可逆地抑制异亮氨酸转移RNA,并抑制细菌蛋白和RNA 的合成起抗菌作用。
T8148 Mupirocin calcium hydrate

莫匹罗星钙,Mupirocin calcium

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Mupirocin calcium hydrate 是从Pseudomonas fluorescens 中分离得到的,一种有口服活性的抗生素。它可逆地抑制异亮氨酸转移RNA,并抑制细菌蛋白和RNA 的合成起到抗菌作用。
TN5466 Boeravinone B

Boeravinone B, a novel efflux pump inhibitor, apart from inhibiting the MdeA mediated efflux, also significantly inhibit the biofilm formation of S. aureus, boeravinone B may be used in combination with mupirocin for further development. Boeravinone B exh

天然产物

Mupirocin
Cat.No: T1465
Synonym: Pseudomonic acid,莫匹罗星,BRL-4910A
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Mupirocin calcium hydrate
Cat.No: T8148
Synonym: 莫匹罗星钙,Mupirocin calcium
Target: Others, Antibacterial, Antibiotic
Boeravinone B
Cat.No: TN5466
Synonym:
Target:
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