Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T68608 |
Methylnaltrexone
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Methylnaltrexone is a narcotic antagonists. | |||
T21422 |
Methylnaltrexone bromide
Relistor,MOA-728,MOA 728,Methylnaltrexone,溴化甲基纳曲酮,MOA728 |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Methylnaltrexone bromide (MOA-728) 是纳曲酮的四元衍生物,是可口服的外周作用 μ 阿片拮抗剂。它穿越血脑屏障的能力有限,可在胃肠道组织中发挥作用。 | |||
T12018 |
Methylnaltrexone-d3 bromide
溴化甲基纳曲酮 D3,Methylnaltrexone D3 Bromide |
Others | Others |
Methylnaltrexone D3 Bromide is the deuterium labeled Methylnaltrexone Bromide. | |||
T40845 |
Methylnaltrexone iodide
Naltrexonium methiodide,碘化甲基纳曲酮; 碘甲纳曲酮 |
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Methylnaltrexone iodide, a quaternary derivative of Naltrexone, is an orally active and selective antagonist of the mu-opioid receptor. It acts peripherally in the gastrointestinal tract to antagonize the receptor. Furthermore, Methylnaltrexone iodide exhibits limited permeability across the blood-brain barrier. | |||
T68358 |
(R)-Methylnaltrexone
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Methylnaltrexone is a narcotic antagonist. |