Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T69134 | Metanicotine | ||
Metanicotine is a selective nicotinic agonist with antinociceptive properties. | |||
T77676 |
(Z)-Metanicotine 2HCl
(Z)-Metanicotine 2HCl(1129-68-6 Free base) |
Others | Others |
(Z)-Metanicotine 2HCl 具有镇痛活性,可用于治疗中枢系统疾病。 | |||
T12738L |
Rivanicline
RJR-2403,(E)-Metanicotine |
Others | Others |
Rivanicline is a neuronal nicotinic receptor agonist, showing high selectivity for the α4β2 subtype (Ki=26 nM). It show > 1,000 fold selectivity than α7 receptors(Ki= 36000 nM and IC50 : 26 nM). | |||
T12739 |
Rivanicline oxalate
RJR-2403 oxalate,(E)-Metanicotine oxalate |
Others | Others |
Rivanicline oxalate is an agonist of neuronal nicotinic receptor, showing high selectivity for the α4β2 subtype (Ki=26 nM). | |||
T12738 |
Rivanicline hemioxalate
RJR-2403 hemioxalate,(E)-Metanicotine hemioxalate |
Others | Others |
Rivanicline hemioxalate (RJR-2403 hemioxalate; (E)-Metanicotine hemioxalate) 是一种神经元烟碱受体 (neuronal nicotinic receptor) 激动剂,对 α4β2 亚型有高度选择性(Ki= 26 nM),比对于 α7 受体的选择性高1000倍(Ki=3.6 μM)。 | |||
T26096 |
RJR-2403 oxalate
RJR 2403 oxalate,Rivanicline oxalate,TC-2403,Metanicotine |
||
RJR-2403 oxalate is a highly selective agonist of α4β2 subtype nicotinic receptor. |