Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T24451 |
Mepyramine
NSC-13136,NSC13136,NSC 13136 |
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Mepyramine is a histamine H1 antagonist. It has mild hypnotic properties and some local anesthetic action and is used for allergies both parenterally and locally. | |||
T1232 |
Mepyramine maleate
马来酸吡纳明,Pyrilamine maleate,吡拉明马来酸盐 |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Mepyramine maleate (Pyrilamine maleate) 是一种组胺 H1 拮抗剂,对 H1、H2 和 H3 受体的 Kd 值分别为 0.8、5200 和大于 3000 nM,对 H1 受体的 pKd 值为 9.4。它是感冒药的常见成分,具有温和的催眠特性和局部麻醉作用,可用于胃肠外和局部过敏。 |