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11

抑制剂 & 化合物

3

天然产物

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Cat. No. Product Name Target Signaling Pathways
T18888 4-Methylumbelliferyl phosphate

4-甲基伞形酮磷酸酯,4-MUP

Others Others
4-Methylumbelliferyl phosphate (4-MUP) 是碱性磷酸酶的荧光底物。
T31458 DiFMUP

DiFMUP is the fluorescent substrate of protein tyrosine phosphatase.
T76735 Mupadolimab

CPI-006

CD73 Immunology/Inflammation
Mupadolimab (CPI-006) 是一种人源化 FcγR 结合缺陷型 IgG1 抗 CD73抗体,具有潜在的抗癌活性,可激活 CD73POS B 细胞。
T25705 Imupedone

LF1695,LF-1695,LF 1695

Others Others
Imupedone (LF 1695) 是一种合成免疫调节剂,可调节 T 淋巴细胞和巨噬细胞,诱导骨髓前体细胞的 T 细胞分化,增加淋巴细胞对有丝分裂原、抗原和同种异体细胞的增殖反应。
TP1473 Velmupressin

c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2

c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 is a selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07nM and 0.02 nM for hV2R and rV2R, respectively.
T75304 Mupirocin calcium

Mupirocin (BRL-4910A, Pseudomonic acid) calcium 可从Pseudomonas fluorescens 中分离得到,是一种有口服活性的抗生素。Mupirocin calcium 通过可逆地抑制异亮氨酸转移 RNA,从而抑制细菌蛋白和 RNA 的合成而发挥抗菌作用。
TP1205 Velmupressin acetate

V2 receptor (V2R) agonist,c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate

c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate is a potent, selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07 and 0.02 nM for hV2R and rV2R, respectively.
T73564 DMUP

DMUP 是一种有效的 CD47-SIRPα axis 抑制剂。DMUP 在 A549 细胞中诱导细胞凋亡 (apoptosis) 并增加巨噬细胞的吞噬作用。DMUP 降低 CD47 和 SIRPα 的蛋白表达水平。DMUP 显示出抗肿瘤活性。
T32406 KMUP-4

KMUP 4

Kmup-4 is an enhancer of cGMP activity and an aortic smooth muscle relaxant.
T32405 KMUP-3

KMUP 3,KMUP3

KMUP-3 is an enhancer of cGMP activity, and acts as an aortic smooth muscle relaxant.
T75340 4-Methylumbelliferyl phosphate disodium

4-Methylumbelliferyl phosphate disodium (4-MUP) 是一种阴离子有机磷酸酯,作为酸性和碱性磷酸酶(phosphatase)的荧光底物,同时也用作神经毒剂模拟剂。

化合物

4-Methylumbelliferyl phosphate
Cat.No: T18888
Synonym: 4-甲基伞形酮磷酸酯,4-MUP
Target: Others
DiFMUP
Cat.No: T31458
Synonym:
Target:
Mupadolimab
Cat.No: T76735
Synonym: CPI-006
Target: CD73
Imupedone
Cat.No: T25705
Synonym: LF1695,LF-1695,LF 1695
Target: Others
Velmupressin
Cat.No: TP1473
Synonym: c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2
Target:
Mupirocin calcium
Cat.No: T75304
Synonym:
Target:
Velmupressin acetate
Cat.No: TP1205
Synonym: V2 receptor (V2R) agonist,c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate
Target:
DMUP
Cat.No: T73564
Synonym:
Target:
KMUP-4
Cat.No: T32406
Synonym: KMUP 4
Target:
KMUP-3
Cat.No: T32405
Synonym: KMUP 3,KMUP3
Target:
4-Methylumbelliferyl phosphate disodium
Cat.No: T75340
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T1465 Mupirocin

Pseudomonic acid,莫匹罗星,BRL-4910A

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Mupirocin (BRL-4910A) 是从Pseudomonas fluorescens 中分离得到的一种有口服活性的抗生素。它可逆地抑制异亮氨酸转移RNA,并抑制细菌蛋白和RNA 的合成起抗菌作用。
T8148 Mupirocin calcium hydrate

莫匹罗星钙,Mupirocin calcium

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Mupirocin calcium hydrate 是从Pseudomonas fluorescens 中分离得到的,一种有口服活性的抗生素。它可逆地抑制异亮氨酸转移RNA,并抑制细菌蛋白和RNA 的合成起到抗菌作用。
TN5951 Mupinensisone

Mupinensisone是一种天然产物,属于卫矛科南蛇藤属,其产品编号为 TN5951,CAS号为 152253-67-3。Mupinensisone可用作对照参考。

天然产物

Mupirocin
Cat.No: T1465
Synonym: Pseudomonic acid,莫匹罗星,BRL-4910A
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Mupirocin calcium hydrate
Cat.No: T8148
Synonym: 莫匹罗星钙,Mupirocin calcium
Target: Others, Antibacterial, Antibiotic
Mupinensisone
Cat.No: TN5951
Synonym:
Target:
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