Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T41247 |
Thioperamide maleate
MR-12842 maleate,硫丙咪胺马来酸 |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Thioperamide maleate (MR-12842 maleate) 是一种有效且选择性的 H3 受体拮抗剂 (Ki = 4.3 nM),可抑制 [3H]histamine 的合成 (Ki = 31 nM)。 | |||
T23456 |
Thioperamide
|
Others | Others |
histamine H3 and H4 antagonist/inverse agonist |