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Cat. No. Product Name Target Signaling Pathways
T6894 ML264

CID-51003603

DNA/RNA Synthesis; KLF Cell Cycle/Checkpoint; DNA Damage/DNA Repair; MAPK
ML264 (CID-51003603) 是抗肿瘤剂,能够特异性地抑制 Krüppel 样因子 5 表达。
T9307 (E)-3-(3,4-dichlorophenyl)-N-(2-(4-(methylsulfonyl)piperazin-1-yl)-2-oxoethyl)acrylamide

Others Others
SR18662 又名 SR18662 ,是一种KLF5 抑制剂, 基于ML264结构的优化而得。它在体内外抑制结直肠癌的生长。
T22429 SR18662

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
SR18662 是 ML264 类似物,可抑制 Krüppel 样因子 5 (KLF5),IC50 为 4.4 nM,降低多种结直肠癌细胞系的活力并诱导细胞凋亡。
T29172 YD277

YD 277,YD-277

YD277 is a small molecule derived from ML264, a KLF5 inhibitor that elicits cytotoxic effects in colon cancer cell lines. YD277 significantly induced G1 cell cycle arrest and apoptosis in MDA-MB-231 and MDA-MB-468 TNBC cells, independent of KLF5 inhibitio

化合物

ML264
Cat.No: T6894
Synonym: CID-51003603
Target: DNA/RNA Synthesis, KLF
(E)-3-(3,4-dichlorophenyl)-N-(2-(4-(methylsulfonyl)piperazin-1-yl)-2-oxoethyl)acrylamide
Cat.No: T9307
Synonym:
Target: Others
SR18662
Cat.No: T22429
Synonym:
Target: DNA/RNA Synthesis
YD277
Cat.No: T29172
Synonym: YD 277,YD-277
Target:
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