Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T12076L |
ML218
|
Calcium Channel | Membrane transporter/Ion channel; Metabolism |
ML218 是一种具有口服活性、选择性、高效性且可穿透血脑屏障的 T 型 Ca2+ 通道抑制剂(Cav3.2 和 Cav3.3 的 IC50 分别为 310 nM 和 270 nM)。ML218 可抑制丘脑下核(STN)神经元的突发性活动。 | |||
T12076 |
ML218 hydrochloride
|
Others | Others |
ML218 hydrochloride is a selective and orally active T-type Ca2+ channels (Cav3.1, Cav3.2, Cav3.3) inhibitor (Cav3.2 and Cav3.3 with IC50s of 310 nM and 270 nM , respectively). |