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Cat. No. Product Name Target Signaling Pathways
T16113 ML753286

AMPK Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
ML753286 has high permeability and low to medium clearance in rodent and human liver S9 fractions. ML753286 is an orally active and selective inhibitor of BCRP (IC50: 0.6 μM). It is also stable in plasma across species.
T10490 (S)-ML753286

Others Others
(S)-ML753286 is a breast cancer resistance protein (BCRP) inhibitor (IC50: 0.6 μM on BCRP efflux transporter).

化合物

ML753286
Cat.No: T16113
Synonym:
Target: AMPK
(S)-ML753286
Cat.No: T10490
Synonym:
Target: Others
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