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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T38163 ML-148

Dehydrogenase Metabolism
ML-148 是 15-羟基前列腺素脱氢酶 (15-PGDH, IC50 = 56 nM) 的特异性抑制剂。 ML-148 可用于分析一组相关的脱氢酶或还原酶以及有关前列腺素信号通路的研究。

化合物

ML-148
Cat.No: T38163
Synonym:
Target: Dehydrogenase
Cat. No. Product Name Target Signaling Pathways
T36329 Terpendole I

Terpendole I is a fungal metabolite that has been found in A. yamanashiensis.1 It is a weak inhibitor of acyl-coenzyme A:cholesterol acyltransferase (ACAT; IC50 = 145 μM) and is active against the bacteria B. cereus and B. subtilis (MICs = 100 μg/ml for both) but not S. aureus, P. aeruginosa, or K. pneumoniae (MICs = >200 μg/ml for all) or the fungus C. albicans (MIC = 200 μg/ml).1,2 It is cytotoxic to HeLa cells with an IC50 value of 52.6 μM.3 |1. Tomoda, H., Tabata, N., Yang, D.-J., et al. Ter...

天然产物

Terpendole I
Cat.No: T36329
Synonym:
Target:
TargetMol Loading
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