Cat. No. | Product Name | Target | Signaling Pathways |
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T70467 |
Alinastine
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Alinastine is a noncompetitive histamine H1 receptor antagonist. | |||
T69952 |
BiBET
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BiBET is a potent, selective, bivalent inhibitor of BET bromodomains. | |||
T70468 |
MK-8666
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MK-8666 is a partial GPCR (G-protein-coupled receptor) agonist that is coordinated with the action of GPR40. GPR40, also known as free fatty acid (FFA) receptor 1 modulates fatty acid-induced insulin secretion in pancreatic beta cells and in intestinal enteroendocrine cells. Thus, MK-8666 has been investigated for treatment of type 2 diabetes mellitus and has been shown to robustly lower glucose without negative effects. |