Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T21456 |
Grazoprevir hydrate
Grazoprevir,MK5172,MK 5172,MK-5172 |
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Grazoprevir, a second generation hepatitis C virus protease inhibitor acting at the NS3/4a protease targets, has good activity against a range of hepatitis C virus genotype variants, including some that are resistant to most currently used antiviral medic | |||
T4547 |
Grazoprevir
MK-5172 |
HCV Protease; SARS-CoV | Microbiology/Virology; Proteases/Proteasome |
Grazoprevir (MK-5172) 是一种丙型肝炎病毒 NS3/4a 蛋白酶的选择性抑制剂,具有跨基因型和耐药变体的广泛活性,对 gt1b、gt1a、gt2a、gt2b 和 gt3a 的Ki 分别为 0.01 nM、0.01 nM、0.08 nM、0.15 nM 和 0.90 nM。它也是 SARS-CoV-2 3CLpro 抑制剂。 | |||
T19948 |
Grazoprevir potassium salt
MK 5172 potassium,Grazoprevir,Grazoprevir potassium,MK 5172,MK5172,MK-5172 |
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Grazoprevir is a drug approved for the treatment of hepatitis C. Grazoprevir is a second-generation hepatitis C virus protease inhibitor acting at the NS3/4a protease targets. | |||
T12065 |
Grazoprevir sodium salt
MK-5172 (sodium salt) |
Others | Others |
Grazoprevir sodium salt is a selective Hepatitis C virus NS3/4a protease inhibitor with broad activity across genotypes and resistant variants. |