Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4442 |
MK2-IN-1 hydrochloride
MK2 Inhibitor,MK 25 |
MAPK | MAPK |
MK2-IN-1 hydrochloride (MK 25) 是一种高效的选择性 MAPKAPK2(MK2)激酶抑制剂,其 IC50值为0.11uM。 | |||
T2126 | MK-5046 | Bombesin Receptor | GPCR/G Protein |
MK5046是一种新型 BRS-3激动剂,同BRS-3结合 (鼠 Ki = 1.6 nM, 人 Ki = 25 nM)的亲和力高。 |