Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T12054L |
MK-0249 FA
MK-0249 FA(862309-06-6 Free base) |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
MK-0249 FA 是一种具有口服活性、选择性和高效性的组胺 H3 反向激动剂,可用于研究成人注意力缺陷、多动症神经分裂和认知障碍。 | |||
T12054 | MK-0249 | Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM). |