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Cat. No. Product Name Target Signaling Pathways
T12475 PIM447

LGH447

Others Others
PIM447 is a potent, orally available, and selective inhibitor of pan-PIM kinase(PIM1, PIM2, and PIM3 with Ki values of 6, 18, and 9 pM , respectively).
T12473 PIM-447 dihydrochloride

LGH447 dihydrochloride

Others Others
PIM-447 dihydrochloride is an orally available and selective inhibitor of pan-PIM kinase(Ki values of 6, 18, and 9 pM for PIM1, PIM2, and PIM3, respectively).
T13425 (1S,3R,5R)-PIM447 dihydrochloride

(1S,3R,5R)-LGH447 dihydrochloride

CDK Cell Cycle/Checkpoint
(1S,3R,5R)-PIM447 (dihydrochloride) an inhibitor of PIM(IC50 of 0.095 μM for Pim1, 0.522 μM for Pim2 and 0.369 μM for Pim3).

化合物

PIM447
Cat.No: T12475
Synonym: LGH447
Target: Others
PIM-447 dihydrochloride
Cat.No: T12473
Synonym: LGH447 dihydrochloride
Target: Others
(1S,3R,5R)-PIM447 dihydrochloride
Cat.No: T13425
Synonym: (1S,3R,5R)-LGH447 dihydrochloride
Target: CDK
TargetMol Loading
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