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3

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T14327 AS1949490

Phosphatase Metabolism
AS1949490 是选择性SHIP-2抑制剂,其IC50=620 nM。它能够通过上调L6肌管GLUT1基因激活葡萄糖代谢。
T67893 PTP1B-IN-22

Phosphatase Metabolism
PTP1B-IN-22是一种蛋白酪氨酸磷酸酶1B (PTP1B)抑制剂,可抑制骨骼肌 L6肌管的葡萄糖摄取。
T25111 AS1938909

AS 1938909,AS-1938909

AS1938909 is a SHIP2 inhibitor that works by increasing Akt phosphorylation, glucose consumption, and glucose uptake in L6 myotubes, specifically upregulating the GLUT1 gene.

化合物

AS1949490
Cat.No: T14327
Synonym:
Target: Phosphatase
PTP1B-IN-22
Cat.No: T67893
Synonym:
Target: Phosphatase
AS1938909
Cat.No: T25111
Synonym: AS 1938909,AS-1938909
Target:
Cat. No. Product Name Target Signaling Pathways
T74199 Beauverolide Ka

Beauverolide Ka 是一种环四缩酚肽,是 Beauveria bassiana 真菌的代谢产物。Beauverolide Ka 浓度为 50 μM 时可刺激培养的大鼠 L6 成肌细胞的葡萄糖摄取。Beauverolide Ka 在 10 μM 时表现出对 HEI-OC1 细胞的保护作用,并且在 L6 成肌细胞和肌管中表现出剂量依赖性活性。
T35532 Galegine hydrochloride

Galegine hydrochloride, a guanidine derivative derived from G. officinalis, plays a role in inducing weight loss in mice and has contributed to the development of biguanides, including metformin and phenformin. This compound stimulates AMPK activation in 3T3-L1 adipocytes, L6 myotubes, H4IIE rat hepatoma, and HEK293 human kidney cell lines. Additionally, galegine hydrochloride exhibits antibacterial properties, particularly demonstrating a minimum inhibitory concentration of 4 mg/L against Staph...

天然产物

Beauverolide Ka
Cat.No: T74199
Synonym:
Target:
Galegine hydrochloride
Cat.No: T35532
Synonym:
Target:
TargetMol Loading
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