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Cat. No. Product Name Target Signaling Pathways
T11752 Keap1-Nrf2-IN-1

Keap1Nrf2-IN-1

Src Angiogenesis; Tyrosine Kinase/Adaptors
Keap1Nrf2 IN-1 activates Nrf2-regulated cytoprotective response and antagonizes acetaminophen-induced liver injury both in cellular and in vivo models. Keap1Nrf2 IN-1 is a Kelch-like ECH-associated protein 1-nuclear factor erythroid 2-related factor 2 (
T64218 Keap1-Nrf2-IN-1 TFA

Keap1-Nrf2-IN-1 TFA (compound35) 是一种 Keap1-Nrf2 蛋白-蛋白相互作用抑制剂 (IC50: 43 nM),可以激活 Nrf2 调节的细胞保护反应。在细胞和体内模型中。Keap1-Nrf2-IN-1 TFA 能够拮抗对乙酰氨基酚诱导的肝损伤。

化合物

Keap1-Nrf2-IN-1
Cat.No: T11752
Synonym: Keap1Nrf2-IN-1
Target: Src
Keap1-Nrf2-IN-1 TFA
Cat.No: T64218
Synonym:
Target:
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