Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11780 |
KRAS G12C inhibitor 5
|
Ras | GPCR/G Protein; MAPK |
KRAS G12C inhibitor 5 is a KRas G12C inhibitor. | |||
T79799 |
pan-KRAS-IN-4
|
Ras | GPCR/G Protein; MAPK |
Pan-KRAS-IN-4 (compound 5) 为一种高效KRAS抑制剂,其IC50值分别为0.37 nM (Kras G12C) 和0.19 nM (Kras G12V)。 | |||
T63164 | KRAS inhibitor-13 | ||
KRAS inhibitor-13 (compound 5-6) 是一种 KRAS G12C 的有效抑制剂 (IC50: 0.883 μM)。KRAS inhibitor-13 在 MIA PaCA-2,A549 细胞中具有 p-ERK 抑制效果,其 IC50 值分别为 5.9,>100 μM。 KRAS inhibitor-13 具有潜力进行胰腺癌、结直肠癌和肺癌的研究。 |