Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T15660 |
KHK-IN-1
KHK-IN-8,Ketohexokinase inhibitor 8 |
Others | Others |
KHK-IN-1 (KHK-IN-8) 是一种选择性的、细胞膜渗透性的己酮糖激酶 (KHK) 抑制剂 (IC50=12 nM; F=34%)。KHK-IN-1 抑制 HepG2 细胞裂解液中 F1P 生成,IC50为400 nM。KHK-IN-1 可用于研究糖尿病和肥胖症。 | |||
T15659 |
KHK-IN-1 hydrochloride
|
Others | Others |
KHK-IN-1 hydrochloride is a potent inhibitor of ketohexokinase (KHK) (IC50: 12 nM). In the ATP-binding region of KHK, KHK-IN-1 hydrochloride interacts with Asp-27B. | |||
T81982 |
KHK-IN-4
|
||
KHK-IN-4(compound 14)是一种针对酮己糖激酶(KHK)的高效抑制剂,适用于果糖代谢疾病的研究。 |