Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T15650 |
KDM5A-IN-1
|
Histone Demethylase | Chromatin/Epigenetic |
KDM5A-IN-1 是一种可口服且具有高效性和选择性的泛组氨酸赖氨酸脱甲基酶 5 KDM5 抑制剂,抑制 KDM5A,KDM5B,KDM5C,IC50 值分别为 45 nM,56 nM 和 55 nM。KDM5A-IN-1 抑制 PC9 H3K4Me3,可用于研究癌症。 | |||
T22299 | CPI-455 HCl | Histone Demethylase | Chromatin/Epigenetic |
CPI-455 is a specific KDM5 inhibitor with IC50 value of 10 ± 1 nM for full-length KDM5A in enzymatic assays, elevating global levels of H3K4 trimethylation (H3K4me3) and decreased the number of DTPs in multiple cancer cell line models treated with target | |||
T73849 | KDM5-C49 hydrochloride | ||
KDM5-C49 (KDOAM-20) hydrochloride 是一种有效和选择性的KDM5去甲基化酶抑制剂,抑制KDM5A,KDM5B 和KDM5C 的IC50值分别为 40 nM,160 nM 和 100 nM。KDM5-C49 hydrochloride 可用于癌症的研究。 |