Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T15638 |
K-252c
|
PKC | Chromatin/Epigenetic; Cytoskeletal Signaling |
K-252c is a staurosporine analog isolated from Nocardiopsis sp. and is a cell-permeable PKC inhibitor (IC50: 2.45 μM). K-252c also inhibits β-lactamase, chymotrypsin, and malate dehydrogenase. K-252c causes apoptosis in human chronic myelogenous leukemia cancer cells. |