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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T3598 JNK-IN-7

JNK inhibitor

JNK MAPK
JNK-IN-7 (JNK inhibitor) 是 JNK 抑制剂,抑制 JNK1、JNK2和 JNK3,IC50分别为 1.5、2 和 0.7 nM。

化合物

JNK-IN-7
Cat.No: T3598
Synonym: JNK inhibitor
Target: JNK
Cat. No. Product Name Target Signaling Pathways
T37452 Stephacidin B

Stephacidin B is a fungal metabolite that has been found inA. ochraceus.1Dimeric stephacidin B is rapidly converted to a monomer, avrainvillamide ,in vitro.2Stephacidin B is cytotoxic to a variety of cancer cells, including testosterone-independent PC3 and -sensitive LNCaP prostate cancer cells (IC50s = 0.37 and 0.06 μM, respectively) and estradiol-independent SK-BR-3 and -sensitive MCF-7 breast cancer cells (IC50s = 0.32 and 0.27 μM, respectively).1It induces apoptosis in HepG2 and Huh7 hepatoc...

天然产物

Stephacidin B
Cat.No: T37452
Synonym:
Target:
TargetMol Loading
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