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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T2057 BVT 2733

Dehydrogenase Metabolism
BVT 2733 是具有口服活性的、强效的、非甾体类11β-HSD1选择性抑制剂。它对小鼠 11β-HSD1 酶的作用 (IC50:96 nM) 比对人 11β-HSD1 酶 (IC50:3341 nM) 的作用强。它对关节炎和肥胖相关疾病具有潜在的研究价值。

化合物

BVT 2733
Cat.No: T2057
Synonym:
Target: Dehydrogenase
Cat. No. Product Name Target Signaling Pathways
TN4050 Fargesone A

NOS Immunology/Inflammation
Fargesone A shows inhibitory effects on nitric oxide (NO) production in the lipopolysaccharide plus interferon-gamma activated-murine macrophage cell line, J774.1.
TN3869 Dimeric coniferyl acetate

Others Others
Dimeric coniferyl acetate has anti-inflammary activity, it shows strong NO inhibition with IC50 values of 27.1 uM in lipopolysacchalide (LPS)-activated murine macrophage-like J774.1 cells. It exhibits significant inhibitory effects on the nitric oxide pro

天然产物

Fargesone A
Cat.No: TN4050
Synonym:
Target: NOS
Dimeric coniferyl acetate
Cat.No: TN3869
Synonym:
Target: Others
TargetMol Loading
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