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Cat. No. Product Name Target Signaling Pathways
T63014 Ivabradine

Ivabradine 是一种有效的、口服具有活力的 HCN (超极化激活的环核苷酸门控) 通道阻滞剂,能够抑制心脏起搏器电流 (If)。Ivabradine 以剂量依赖性的方式降低心率,且不改变血压。Ivabradine 具有抗惊厥、抗缺血和抗心绞痛作用。
T2535 Ivabradine hydrochloride

盐酸伊伐布雷定,S 16257-2,Ivabradine HCl

Adrenergic Receptor GPCR/G Protein; Neuroscience
Ivabradine hydrochloride (S 16257-2) 是一种可口服的,超极化激活的环核苷酸门控离子通道通道阻滞剂。
T11695 N-Demethyl ivabradine hydrochloride

Ivabradine metabolite N-Demethyl Ivabradine hydrochloride

Others Others
N-Demethyl Ivabradine Hcl is a specific inhibitor of the funny channel.N-Demethyl Ivabradine Hcl is a metabolite of Ivabradine.
T11694 Ivabradine-d6 hydrochloride

盐酸伊伐布雷定 D6,Ivabradine D6 hydrochloride

Others Others
Ivabradine hydrochloride is a new If inhibitor with IC50 of 2.9 μM, and used as a pure heart rate lowering agent. Ivabradine D6 hydrochloride is the deuterium labeled Ivabradine hydrochloride.
T37160 8-Demethyl Ivabradine

8-Demethyl Ivabradine is a metabolite derived from Ivabradine, an orally bioavailable cyclic nucleotide-gated (HCN) channel blocker with hyperpolarization-activated properties[1].
T11692 Ivabradine-d3 hydrochloride

盐酸伊伐布雷定 D3,Ivabradine D3 Hydrochloride

Others Others
Ivabradine hydrochloride is a new If inhibitor with IC50 of 2.9 μM, and used as a pure heart rate lowering agent. Ivabradine D3 Hydrochloride is the deuterium labeled Ivabradine hydrochloride.
T19447 N-Demethyl Ivabradine D6 Hydrochloride

Others Others
N-Demethyl Ivabradine D6 Hydrochloride salt is the deuterium labeled N-Demethyl Ivabradine, which is a Ivabradine metabolite.
T73976 Ivabradine impurity 2

Ivabradine impurity 2 是 Ivabradine 的一个杂质。 Ivabradine 是具有口服活性的,超极化激活的环核苷酸门控离子通道 (HCN) 通道阻滞剂。
T73975 Ivabradine impurity 1

Ivabradine impurity 1 是Ivabradine 的一个杂质。 Ivabradine 是具有口服活性的,超极化激活的环核苷酸门控离子通道 (HCN) 通道阻滞剂。

化合物

Ivabradine
Cat.No: T63014
Synonym:
Target:
Ivabradine hydrochloride
Cat.No: T2535
Synonym: 盐酸伊伐布雷定,S 16257-2,Ivabradine HCl
Target: Adrenergic Receptor
N-Demethyl ivabradine hydrochloride
Cat.No: T11695
Synonym: Ivabradine metabolite N-Demethyl Ivabradine hydrochloride
Target: Others
Ivabradine-d6 hydrochloride
Cat.No: T11694
Synonym: 盐酸伊伐布雷定 D6,Ivabradine D6 hydrochloride
Target: Others
8-Demethyl Ivabradine
Cat.No: T37160
Synonym:
Target:
Ivabradine-d3 hydrochloride
Cat.No: T11692
Synonym: 盐酸伊伐布雷定 D3,Ivabradine D3 Hydrochloride
Target: Others
N-Demethyl Ivabradine D6 Hydrochloride
Cat.No: T19447
Synonym:
Target: Others
Ivabradine impurity 2
Cat.No: T73976
Synonym:
Target:
Ivabradine impurity 1
Cat.No: T73975
Synonym:
Target:
TargetMol Loading
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