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Cat. No. Product Name Target Signaling Pathways
T4986 Imidafenacin

咪达那新,KRP-197,ONO-8025

AChR Neuroscience
Imidafenacin (KRP-197) 是一种有效的和选择性的 M3受体抑制剂,Kb 值为0.317nM。
T36662 Imidafenacin Metabolite M4

Imidafenacin Metabolite M4

Imidafenacin metabolite M4 is a metabolite of the muscarinic acetylcholine receptor antagonist imidafenacin.1It is formed from imidafenacin by the cytochrome P450 (CYP) isoform CYP3A4. 1.Kanayama, N., Kanari, C., Masuda, Y., et al.Drug-drug interactions in the metabolism of imidafenacin: Role of the human cytochrome P450 enzymes and UDP-glucuronic acid transferases, and potential of imidafenacin to inhibit human cytochrome P450 enzymesXenobiotica37(2)139-154(2007)

化合物

Imidafenacin
Cat.No: T4986
Synonym: 咪达那新,KRP-197,ONO-8025
Target: AChR
Imidafenacin Metabolite M4
Cat.No: T36662
Synonym: Imidafenacin Metabolite M4
Target:
TargetMol Loading
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