Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4986 |
Imidafenacin
咪达那新,KRP-197,ONO-8025 |
AChR | Neuroscience |
Imidafenacin (KRP-197) 是一种有效的和选择性的 M3受体抑制剂,Kb 值为0.317nM。 | |||
T36662 |
Imidafenacin Metabolite M4
Imidafenacin Metabolite M4 |
||
Imidafenacin metabolite M4 is a metabolite of the muscarinic acetylcholine receptor antagonist imidafenacin.1It is formed from imidafenacin by the cytochrome P450 (CYP) isoform CYP3A4. 1.Kanayama, N., Kanari, C., Masuda, Y., et al.Drug-drug interactions in the metabolism of imidafenacin: Role of the human cytochrome P450 enzymes and UDP-glucuronic acid transferases, and potential of imidafenacin to inhibit human cytochrome P450 enzymesXenobiotica37(2)139-154(2007) |