Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TQ0016 |
NKP-1339
IT-139,KP-1339 |
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
NKP-1339 (IT-139) induces G2/M cell cycle arrest, blockage of DNA synthesis, and induction of apoptosis via the mitochondrial pathway. | |||
T72543 |
BOLD-100 free base
NKP-1339 free base ; IT-139 free base ; KP-1339 free base,KP-1339 free base,NKP-1339 free base,IT-139 free base |
||
BOLD-100 (NKP-1339; IT-139) free base 是一款钌基抗癌药物。作为GRP78应激诱导上调的抑制剂,它破坏内质网(ER)的稳态,从而诱发ER应激和未折叠蛋白反应(UPR)。此外,BOLD-100 free base 干预了内质网应激反应、溶酶体动力学以及细胞自噬(autophagy)间的复杂交互作用。 |