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Cat. No. Product Name Target Signaling Pathways
T1988 Duvelisib

INK1197,IPI-145,度维利塞

PI3K PI3K/Akt/mTOR signaling
Duvelisib (INK1197) 是 p100δ的选择性抑制剂,能够作用于 p110δ (IC50:2.5 nM)、p110γ (IC50:27.4 nM)、p110β (IC50:85 nM) 和 p110α (IC50:1602 nM)。
T11129L Duvelisib (R enantiomer) hydrochloride

IPI-145 R enantiomer HCl,Duvelisib (R enantiomer) hydrochloride(1261590-48-0 Free base),INK1197 R enantiomer HCl

PI3K PI3K/Akt/mTOR signaling
Duvelisib (R enantiomer) hydrochloride (INK1197 R enantiomer HCl) 是 PI3K 抑制剂。Duvelisib (R enantiomer) hydrochloride 是 Duvelisib 的活性较低的对映体。
T11129 Duvelisib (R enantiomer)

Duvelisib R enantiomer,IPI-145 R enantiomer,INK1197 R enantiomer

PI3K PI3K/Akt/mTOR signaling
Duvelisib R enantiomer (IPI-145 R enantiomer) 是一种 Duvelisib 的对映异构体,活性较低。 它是一种 PI3K 抑制剂。
T70800 Elenbecestat free base

Elenbecestat,also known as E2609 is a BACE1 inhibitor. By inhibiting BACE, a key enzyme in the production of Aβ peptides, E2609 decreases the formation of these peptides which can aggregate into toxic oligomers and protofibrils and eventually form amyloid plaques in the brain. Elenbecestat has been shown to reduce Aβ levels in cerebrospinal fluid, was investigated in two global phase 3 studies in early AD.

化合物

Duvelisib
Cat.No: T1988
Synonym: INK1197,IPI-145,度维利塞
Target: PI3K
Duvelisib (R enantiomer) hydrochloride
Cat.No: T11129L
Synonym: IPI-145 R enantiomer HCl,Duvelisib (R enantiomer) hydrochloride(1261590-48-0 Free base),INK1197 R enantiomer HCl
Target: PI3K
Duvelisib (R enantiomer)
Cat.No: T11129
Synonym: Duvelisib R enantiomer,IPI-145 R enantiomer,INK1197 R enantiomer
Target: PI3K
Elenbecestat free base
Cat.No: T70800
Synonym:
Target:
TargetMol Loading
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